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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5480 | BI-4464 | FAK , Ligands for Target Protein for PROTAC | |
BI-4464 is a highly selective ATP competitive inhibitor of PTK2/FAK, with an IC50 of 17 nM. A PTK2 ligand for PROTAC | |||
T17543 | BI-3663 | Others | |
BI-3663 is a highly selective PTK2/FAK PROTAC, with cereblon ligands to hijack E3 ligases for PTK2 degradation. BI-3663 inhibits PTK2 with an IC50 of 18 nM. BI-3663 is a PROTAC that composes of BI-4464 linked to Pomalido... |